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Page values for "Exenatide"

From Pharmacopedia
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"Medicines" values

1 row is stored for this page
FieldField typeValue
genericStringExenatide
brandStringByetta (twice-daily), Bydureon BCise (weekly)
structureFile
classesList of String, delimiter: ,[[GLP-1 receptor agonist]] · [[Antidiabetic medicines|Antidiabetic]] · First-in-class incretin mimetic
mechanismStringAgonist of the [[GLP-1 receptor]]; exendin-4 derivative from Gila monster venom.
usesString[[Type 2 diabetes mellitus]] (adjunct, second-line)
starting_doseStringByetta: 5 µg SC twice daily, within 60 min before morning and evening meals'"`UNIQ--ref-000000E3-QINU`"' · Bydureon BCise: 2 mg SC once weekly'"`UNIQ--ref-000000E4-QINU`"'
preparationsStringByetta pre-filled multi-dose pen: 5 µg / 10 µg per dose'"`UNIQ--ref-000000E5-QINU`"' · Bydureon BCise single-dose autoinjector: 2 mg extended-release microsphere suspension'"`UNIQ--ref-000000E6-QINU`"'
fda_maxString10 µg twice daily (Byetta)'"`UNIQ--ref-000000E7-QINU`"' · 2 mg once weekly (Bydureon BCise)'"`UNIQ--ref-000000E8-QINU`"'
pill_idText
routesList of String, delimiter: ,Subcutaneous (abdomen thigh upper arm)'"`UNIQ--ref-000000E9-QINU`"'
onsetStringGlycemic effect within hours (Byetta); weeks (Bydureon, extended-release microsphere)'"`UNIQ--ref-000000EA-QINU`"'
durationString~10 hours (Byetta)'"`UNIQ--ref-000000EB-QINU`"' · ~7 days steady-state (Bydureon, after ~6–7 weeks of weekly dosing to reach steady state)'"`UNIQ--ref-000000EC-QINU`"'
halflifeString~2.4 hours (Byetta, short, hence the BID schedule)'"`UNIQ--ref-000000ED-QINU`"' · Effective release half-life ~2 weeks (Bydureon)'"`UNIQ--ref-000000EE-QINU`"'
bioavailabilityStringSC ~65%–75%<sup class="pcp-cn" title="This claim needs a citation.">&#91;[[Pharmacopedia:Citation needed|citation&nbsp;needed]]&#93;</sup>
pregnancyStringAvoid. Discontinue before planned pregnancy.'"`UNIQ--ref-000000EF-QINU`"'
legalStringRx-only;'"`UNIQ--ref-000000F0-QINU`"' not a controlled substance