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Page values for "Sitagliptin"

From Pharmacopedia
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"Medicines" values

1 row is stored for this page
FieldField typeValue
genericStringSitagliptin
brandStringJanuvia; with metformin Janumet/Janumet XR
structureFile
classesList of String, delimiter: ,[[:Category:DPP-4_inhibitors|DPP-4 inhibitor]] [[:Category:Antihyperglycemic_agents|Antihyperglycemic agent]] [[:Category:Incretin_modulators|Incretin pathway modulator]]
mechanismString'"`UNIQ--vote-00000762-QINU`"' Largely renally cleared, hence the eGFR-tiered dosing. Rare but well-documented signals: acute pancreatitis (uncertain causal contribution), severe joint pain, and bullous pemphigoid (class effect, especially in older Asian patients)'"`UNIQ--ref-00000763-QINU`"'.
usesString'"`UNIQ--vote-00000764-QINU`"'
starting_doseString100 mg PO once daily (50 mg if CrCl 30-44; 25 mg if <30 or dialysis)
preparationsString25, 50, 100 mg tablets; combination tablets with metformin
fda_maxString100 mg/d
pill_idText
routesList of String, delimiter: ,Oral
onsetStringPostprandial glucose effect within days; HbA1c by 12 weeks
durationString24 hours
halflifeString~12.4 hours'"`UNIQ--ref-00000765-QINU`"'
bioavailabilityString~87% (oral)'"`UNIQ--ref-00000766-QINU`"'
pregnancyStringLimited data; switch to insulin where feasible.<sup class="pcp-cn" title="This claim needs a citation.">&#91;[[Pharmacopedia:Citation needed|citation&nbsp;needed]]&#93;</sup>
legalString[[USLegal:Prescription only|Rx-only]] in US