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Methamphetamine: Difference between revisions

From Pharmacopedia
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Pharmacopedia: remove contraindications parameter
Line 50: Line 50:
| pk_elimination    = Urinary elimination is pH-dependent.
| pk_elimination    = Urinary elimination is pH-dependent.
| pharmacodynamics  = Methamphetamine acts at monoaminergic terminals as a releasing agent via TAAR1 agonism, VMAT2 substrate activity, and DAT/NET reverse transport. Secondary mechanisms include weak monoamine reuptake inhibition.
| pharmacodynamics  = Methamphetamine acts at monoaminergic terminals as a releasing agent via TAAR1 agonism, VMAT2 substrate activity, and DAT/NET reverse transport. Secondary mechanisms include weak monoamine reuptake inhibition.
| contraindications = Per Desoxyn label:
* Advanced arteriosclerosis
* Symptomatic cardiovascular disease
* Moderate to severe hypertension
* Hyperthyroidism
* Known hypersensitivity to sympathomimetic amines
* Glaucoma
* Agitated states
* History of drug abuse (per label wording)
* Concurrent MAOI use, or within 14 days of MAOI discontinuation
| interactions      = * '''MAOIs''' — contraindicated (per label)
| interactions      = * '''MAOIs''' — contraindicated (per label)
* '''Acidifying agents''' — increase urinary clearance
* '''Acidifying agents''' — increase urinary clearance