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Tizanidine: Difference between revisions

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Revision as of 03:31, 14 May 2026

Muscle relaxant
Tizanidine
Zanaflex

Experience

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Problems

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Titration strategies

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Effects

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Interactions

Pharmacogenomic + mechanism interactions2 edges
Pharmacokinetic mechanismSubstrate / metabolism relationships from primary literature
Enzyme:CYP1A2 substrate major Primary 80 / 100
FDA Drug Interactions Table: sensitive index substrate of CYP1A2.
Inferred from pharmacokinetic dataMaterialised by the inference engine; provenance shown per row
Fluvoxamine pk raises via CYP1A2 Inferred 72 / 100
Fluvoxamine inhibits CYP1A2 (inhibitor_strong, intensity 90); Tizanidine is a substrate_major of CYP1A2 (intensity 80). Derived: Tizanidine exposure raised.
Inferred via Enzyme:CYP1A2 (exposure raised)

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Relevant Literature

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Summary
Classes
Muscle relaxant
Common uses
Pharmacy
Pharmacology
Purported mechanism
Alpha-2 adrenergic receptor agonist