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Drilldown: Medicines

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Medicines > classes : Cathinone or GABA-A positive allosteric modulator (oral)

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generic:
None (1) · 3-MMC (1) · Butylone (1) · Cathinone (1) · Ephylone (1) · Ethcathinone (1) · Ethylone (1) · Hexedrone (1) · Mephedrone (1) · Methcathinone (1) · Methylone (1) · Mexedrone (1) · N-Ethylhexedrone (1) · N-Ethylpentedrone (1) · Pentedrone (1)
brand:
None (14) · Zurzuvae (1)
classes: (Click arrow to add another value)
mechanism:
Cathinone analogue; monoamine reuptake inhibitor (2) · Monoamine releasing agent (4) · Monoamine releasing agent; active ingredient in khat (1) · Norepinephrine and dopamine releasing agent (1) · Norepinephrine/dopamine releasing agent (1) · Norepinephrine/dopamine reuptake inhibitor (1) · Serotonin releasing agent; monoamine reuptake inhibitor (1) · Serotonin/norepinephrine/dopamine releasing agent (3) · Synthetic neuroactive steroid (an analog of allopregnanolone), bioavailable orally unlike brexanolone. Positive allosteric modulator at GABA-A receptors including extrasynaptic δ-containing subtypes. (1)
uses:
None (14) · Postpartum depression (PPD) in adults (FDA-approved 2023) (1)
starting dose:
None (14) · 50 mg PO once daily with fatty food in the evening × 14 days (1)
preparations:
None (14) · 20 mg, 25 mg, 30 mg capsules (1)
fda max:
None (14) · 50 mg/d × 14 d (1)
routes:
None (14) · Oral (1)
onset:
None (14) · Day 3 of dosing in trials; sustained through day 45 (1)
duration:
None (14) · 14-day course; effect persists after discontinuation in trials (1)
halflife:
None (14) · ~16-23 hours (1)
bioavailability:
None (14) · Adequate (food-dependent, must take with fatty meal) (1)
pregnancy:
None (14) · Limited data; avoid in pregnancy. Lactation: present in milk; consider risks (1)
legal:
None (14) · Rx, Schedule IV (US) (1)

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