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Medicines > classes : Cathinone or GABAB Agonist; Endogenous GHB receptor agonist

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generic:
3-MMC (1) · Butylone (1) · Cathinone (1) · Ephylone (1) · Ethcathinone (1) · Ethylone (1) · Hexedrone (1) · Mephedrone (1) · Methcathinone (1) · Methylone (1) · Mexedrone (1) · N-Ethylhexedrone (1) · N-Ethylpentedrone (1) · Pentedrone (1) · Sodium Oxybate (1)
brand:
None (14) · Xyrem; Xywav (lower-sodium formulation with Ca/Mg/K salts) (1)
classes: (Click arrow to add another value)
mechanism:
Agonist at the metabotropic GABAB receptor and the endogenous γ-hydroxybutyrate (GHB) receptor. Produces deep sleep with increased slow-wave architecture, suppression of REM intrusion, and cataplexy reduction. (1) · Cathinone analogue; monoamine reuptake inhibitor (2) · Monoamine releasing agent (4) · Monoamine releasing agent; active ingredient in khat (1) · Norepinephrine and dopamine releasing agent (1) · Norepinephrine/dopamine releasing agent (1) · Norepinephrine/dopamine reuptake inhibitor (1) · Serotonin releasing agent; monoamine reuptake inhibitor (1) · Serotonin/norepinephrine/dopamine releasing agent (3)
uses:
None (14) · '"`UNIQ--vote-00000717-QINU`"', '"`UNIQ--vote-00000718-QINU`"', '"`UNIQ--vote-00000719-QINU`"' (1)
starting dose:
None (14) · 2.25 g at bedtime + 2.25 g 2.5–4 h later; titrate weekly to 6–9 g/night total (1)
preparations:
None (14) · 0.5 g/mL oral solution (1)
fda max:
None (14) · 9 g/night (1)
routes:
None (14) · Oral (must be taken in bed; effects within minutes) (1)
onset:
None (14) · 15–30 min (fasting) (1)
duration:
None (14) · ~3 h per dose (twice-nightly schedule required) (1)
halflife:
None (14) · 30–60 min (1)
bioavailability:
None (14) · ~25% (high first-pass) (1)
pregnancy:
None (14) · Category C (1)
legal:
None (14) · Schedule III; REMS-restricted (Schedule I if outside the pharmaceutical channel, same molecule as illicit GHB) (1)

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