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Medicines (732)

Medicines > routes: Oral

& duration

: 24 h

or 4–6 h

Use the filters below to narrow your results.

Avanafil (1) · Bisoprolol (1) · Nebivolol (1)

Bystolic (1) · Stendra (1) · Zebeta (1)

Beta Blocker (2) · Cardioselective (β1) (1) · Cardioselective (β1) + vasodilator (1) · PDE5 Inhibitor (1)

Highly β1-selective adrenergic antagonist. Greater selectivity than metoprolol or atenolol. (1) · Selective inhibitor of phosphodiesterase type 5 (PDE5); increases cGMP in cavernous smooth muscle, producing erection in response to sexual stimulation. (1) · The d-enantiomer is a highly β1-selective antagonist; the l-enantiomer triggers endothelial nitric-oxide–mediated vasodilation. Unique among beta blockers for this NO mechanism. (1)

'"`UNIQ--vote-00000040-QINU`"' (1) · '"`UNIQ--vote-0000059D-QINU`"' (1) · '"`UNIQ--vote-00000636-QINU`"', '"`UNIQ--vote-00000637-QINU`"', '"`UNIQ--vote-00000638-QINU`"' (1)

100 mg ~15 min before sexual activity (1) · 2.5–5 mg daily (HTN); 1.25 mg daily (HFrEF, slow titration) (1) · 5 mg daily (1)

2.5, 5, 10, 20 mg tabs (1) · 5, 10 mg tabs (1) · 50, 100, 200 mg tabs (1)

20 mg/d (1) · 200 mg/d (100 mg/d if on CYP3A4 inhibitors) (1) · 40 mg/d (1)

1–2 h (2) · ~15 min (fastest of the PDE5 inhibitors) (1)

9–12 h (1) · ~10 h (CYP2D6 extensive metabolizers); up to 31 h (poor metabolizers) (1) · ~5 h (1)

Rapid absorption; absolute bioavailability not formally established (1) · ~12% (extensive metabolizers); ~96% (poor metabolizers) (1) · ~90% (low first-pass) (1)

Category C (2) · Category C (not relevant; not used in women) (1)

Rx-only in US (3)

Showing below up to 3 results in range #1 to #3.

A

Avanafil

B

Bisoprolol

N

Nebivolol

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