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Medicines (732)

Medicines > routes: Oral

& duration

: 24 h

or IR 3–5 h; LA/SR 6–8 h; Concerta 10–12 h; Daytrana ~9 h wear time

Use the filters below to narrow your results.

Bisoprolol (1) · Methylphenidate (1) · Nebivolol (1)

Bystolic (1) · Ritalin, Ritalin LA, Concerta, Metadate CD, Daytrana, Quillivant XR (1) · Zebeta (1)

Beta Blocker (2) · Cardioselective (β1) (1) · Cardioselective (β1) + vasodilator (1) · NDRI (1) · Psychostimulant (1)

Highly β1-selective adrenergic antagonist. Greater selectivity than metoprolol or atenolol. (1) · Norepinephrine–dopamine reuptake inhibition (DAT, NET) (1) · The d-enantiomer is a highly β1-selective antagonist; the l-enantiomer triggers endothelial nitric-oxide–mediated vasodilation. Unique among beta blockers for this NO mechanism. (1)

ADHD, narcolepsy (1) · '"`UNIQ--vote-0000059D-QINU`"' (1) · '"`UNIQ--vote-00000636-QINU`"', '"`UNIQ--vote-00000637-QINU`"', '"`UNIQ--vote-00000638-QINU`"' (1)

None (1) · 2.5–5 mg daily (HTN); 1.25 mg daily (HFrEF, slow titration) (1) · 5 mg daily (1)

None (1) · 2.5, 5, 10, 20 mg tabs (1) · 5, 10 mg tabs (1)

None (1) · 20 mg/d (1) · 40 mg/d (1)

1–2 h (2) · 20–60 min (oral) (1)

2–3 h (parent compound) (1) · 9–12 h (1) · ~10 h (CYP2D6 extensive metabolizers); up to 31 h (poor metabolizers) (1)

~12% (extensive metabolizers); ~96% (poor metabolizers) (1) · ~30% (high first-pass) (1) · ~90% (low first-pass) (1)

Category C (2) · Pregnancy categories were retired by FDA in 2015. Limited reproductive data with small observational signal for cardiac malformations; risk-benefit decision, with many patients deferring ADHD treatment during pregnancy. See pregnancy_details for the full discussion. (1)

Rx-only in US (2) · Schedule II (1)

Showing below up to 3 results in range #1 to #3.

B

Bisoprolol

M

Methylphenidate

N

Nebivolol

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