Jump to content

Drilldown: Medicines

Choose a table:


Medicines > classes : Cardioselective (β1) + vasodilator or Cathinone or Opioid

Use the filters below to narrow your results.

generic:
Codeine (2)
brand:
None (26) · (multiple, generic dominant) (1) · Alfenta (1) · Bystolic (1) · Darvon (1) · Demerol (1) · Dilaudid (1) · Duragesic (1) · Heroin (1) · Krokodil (1) · Nubain (1) · Nucynta (1) · O-DSMT (1) · Opana (1) · Stablon (1) · Stadol (1) · Sufenta (1) · Talwin (1) · Ultiva (1) · Vicodin (1)
classes: (Click arrow to add another value)
mechanism:
Active metabolite of tramadol; mu-opioid agonist (1) · Cathinone analogue; monoamine reuptake inhibitor (2) · Extremely potent mu-opioid receptor agonist (1) · Highly potent mu-opioid receptor agonist (1) · Kappa agonist; mu antagonist (1) · Kappa agonist; mu partial agonist (1) · Kappa agonist; mu partial agonist/antagonist (1) · Mitragynine/7-hydroxymitragynine; mu-opioid partial agonist (1) · Monoamine releasing agent (4) · Monoamine releasing agent; active ingredient in khat (1) · Mu-opioid agonist; modulates glutamate AMPA receptors (1) · Mu-opioid agonist; norepinephrine reuptake inhibitor (1) · Mu-opioid receptor agonist (4) · Mu-opioid receptor agonist; fentanyl analogue (1) · Mu-opioid receptor agonist; prodrug (metabolized to morphine) (1) · Mu-opioid receptor agonist; sodium channel blocker (1) · Mu/kappa/delta agonist; NMDA antagonist (1) · Norepinephrine and dopamine releasing agent (1) · Norepinephrine/dopamine releasing agent (1) · Norepinephrine/dopamine reuptake inhibitor (1) · Opioid receptor partial agonist/antagonist; toxic alkaloid (1) · Partial mu-opioid receptor agonist; alpha-2 agonist (1) · Phosphodiesterase inhibitor; calcium channel blocker (1) · Potent mu-opioid receptor agonist (6) · Prodrug of morphine; mu-opioid receptor agonist (1) · Prodrug; converted to [[Morphine|morphine]] by [[Enzyme:CYP2D6|CYP2D6]] for analgesic action. (1) · Selective mu-opioid receptor agonist (1) · Serotonin releasing agent; monoamine reuptake inhibitor (1) · Serotonin/norepinephrine/dopamine releasing agent (3) · The d-enantiomer is a highly β1-selective antagonist; the l-enantiomer triggers endothelial nitric-oxide–mediated vasodilation. Unique among beta blockers for this NO mechanism. (1) · Ultra-short-acting mu-opioid agonist (1)
uses:
None (43) · Mild to moderate pain; cough suppression (low-dose). (1) · '"`UNIQ--vote-0000059D-QINU`"' (1)
starting dose:
None (43) · 5 mg daily (1) · Adult: 15–60 mg every 4 hours as needed. (1)
preparations:
None (43) · 2.5, 5, 10, 20 mg tabs (1) · Tablet (15, 30, 60 mg); oral solution; combination products (with [[Acetaminophen|acetaminophen]] or ibuprofen). (1)
fda max:
None (43) · 360 mg/day (1) · 40 mg/d (1)
routes:
None (43) · Oral (1) · PO (only formulation marketed in the US). (1)
onset:
None (43) · 1–2 h (1) · 30–60 min (PO) (1)
duration:
None (43) · 24 h (1) · 4–6 hours (1)
halflife:
None (43) · 2.5–3 hours (1) · ~10 h (CYP2D6 extensive metabolizers); up to 31 h (poor metabolizers) (1)
bioavailability:
None (43) · ~12% (extensive metabolizers); ~96% (poor metabolizers) (1) · ~50% (variable, CYP2D6-dependent for analgesic effect). (1)
pregnancy:
None (43) · Avoid; risk of neonatal opioid withdrawal with chronic use; UM-mother breastfeeding contraindicated. (1) · Category C (1)
legal:
None (43) · Rx-only in US (1) · US Schedule II (single-entity); Schedule III–V (combination products by content). (1)

Showing below up to 45 results in range #1 to #45.

View (previous 250 | next 250) (20 | 50 | 100 | 250 | 500)


View (previous 250 | next 250) (20 | 50 | 100 | 250 | 500)

Retrieved from "https://pharmacopedia.wiki/p/Special:Drilldown/Medicines"